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1

Human M1-, M2- and M3-muscarinic cholinergic receptors: Binding characteristics of agonists and antagonists

Patrick Vanderheyden, Jean-Pierre Gies, Guy Ebinger, Jacques De Keyser, Yves Landry, Georges Vauquelin

Journal:

Journal of the Neurological Sciences

Year:

1990

Language:

english

File:

PDF, 739 KB

english, 1990

2

Radioligand binding to intact cells as a tool for extended drug screening in a representative physiological context

Vauquelin, Georges, Van Liefde, Isabelle, Swinney, David C.

Journal:

Drug Discovery Today: Technologies

Year:

2015

Language:

english

File:

PDF, 692 KB

english, 2015

3

Age-related changes in the human nigrostriatal dopaminergic system

MD Jacques De Keyser, MD Guy Ebinger, MD, PhD Georges Vauquelin

Journal:

Annals of Neurology

Year:

1990

Language:

english

File:

PDF, 513 KB

english, 1990

4

Ligands to the (IRAP)/AT4 receptor encompassing a 4-hydroxydiphenylmethane scaffold replacing Tyr2

Hanna Andersson, Heidi Demaegdt, Georges Vauquelin, Gunnar Lindeberg, Anders Karlén, Mathias Hallberg

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 517 KB

english, 2008

5

Molecular characterization of the high-affinity [3H]neuropeptide Y-binding component from the venom of Conus anemone

Minh Tam Le, Patrick M. L. Vanderheyden, Frederik L. P. Fierens, George Vauquelin

Journal:

Fundamental & Clinical Pharmacology

Year:

2003

Language:

english

File:

PDF, 158 KB

english, 2003

6

Conformational constraints in angiotensin IV to probe the role of Tyr2, Pro5 and Phe6

Aneta Lukaszuk, Heidi Demaegdt, Isabelle Van den Eynde, Patrick Vanderheyden, Georges Vauquelin, Dirk Tourwé

Journal:

Journal of Peptide Science

Year:

2011

Language:

english

File:

PDF, 279 KB

english, 2011

7

Cyclic insulin-regulated aminopeptidase (IRAP)/AT4 receptor ligands

Andreas Axén, Gunnar Lindeberg, Heidi Demaegdt, Georges Vauquelin, Anders Karlén, Mathias Hallberg

Journal:

Journal of Peptide Science

Year:

2006

Language:

english

File:

PDF, 206 KB

english, 2006

8

Small potent ligands to the insulin-regulated aminopeptidase (IRAP)/AT4 receptor

Andreas Axén, Hanna Andersson, Gunnar Lindeberg, Harriet Rönnholm, Jarkko Kortesmaa, Heidi Demaegdt, Georges Vauquelin, Anders Karlén, Mathias Hallberg

Journal:

Journal of Peptide Science

Year:

2007

Language:

english

File:

PDF, 234 KB

english, 2007

9

Evaluation of bioactive saponins and triterpenoidal aglycons for their binding properties on human endothelin ETA and angiotensin AT1 receptors

C. Caballero-George, P. M. L. Vanderheyden, Y. Okamoto, T. Masaki, Z. Mbwambo, S. Apers, M. P. Gupta, L. Pieters, G. Vauquelin, A. Vlietinck

Journal:

Phytotherapy Research

Year:

2004

Language:

english

File:

PDF, 245 KB

english, 2004

10

Involvement of insulin-regulated aminopeptidase in the effects of the renin–angiotensin fragment angiotensin IV: a review

Bart Stragier, Dimitri De Bundel, Sophie Sarre, Ilse Smolders, Georges Vauquelin, Alain Dupont, Yvette Michotte, Patrick Vanderheyden

Journal:

Heart Failure Reviews

Year:

2008

Language:

english

File:

PDF, 366 KB

english, 2008

11

D2 Dopamine Receptors in Calf Globus Pallidus: Agonist High- and Low-Affinity Sites Not Regulated by Guanine Nucleotide

Jacques De Keyser, Jean-Paul De Backer, André Convents, Guy Ebinger, Georges Vauquelin

Journal:

Journal of Neurochemistry

Year:

1985

Language:

english

File:

PDF, 330 KB

english, 1985

12

[3H]GBR 12935 Binding to Dopamine Uptake Sites in the Human Brain

Jacques De Keyser, Jean-Paul De Backer, Guy Ebinger, Georges Vauquelin

Journal:

Journal of Neurochemistry

Year:

1989

Language:

english

File:

PDF, 1011 KB

english, 1989

13

In Human Brain Two Subtypes of D1 Dopamine Receptors Can Be Distinguished on the Basis of Differences in Guanine Nucleotide Effect on Agonist Binding

Jacques de Keyser, Hiljle Walraevens, Guy Ebinger, Georges Vauquelin

Journal:

Journal of Neurochemistry

Year:

1989

Language:

english

File:

PDF, 1.04 MB

english, 1989

14

D1 and D2 Dopamine Receptors in Human Substantia Nigra: Localization and the Effect of Aging

Jacques De Keyser, Jean-Paul De Backer, Georges Vauquelin, Guy Ebinger

Journal:

Journal of Neurochemistry

Year:

1991

Language:

english

File:

PDF, 431 KB

english, 1991

15

Regional Distribution of α2A-and α2B-Adrenoceptor Subtypes in Postmortem Human Brain

Hilde De Vos, Georges Vauquelin, Jacques De Keyser, Jean-Paul De Backer, Isabelle Van Liefde

Journal:

Journal of Neurochemistry

Year:

1992

Language:

english

File:

PDF, 612 KB

english, 1992

16

Metabolism of angiotensin II is required for its in vivo effect on dopamine release in the striatum of the rat

Bart Stragier, Sophie Sarre, Patrick Vanderheyden, Georges Vauquelin, Marie-Claude Fournié-Zaluski, Guy Ebinger, Yvette Michotte

Journal:

Journal of Neurochemistry

Year:

2004

Language:

english

File:

PDF, 161 KB

english, 2004

17

Expression, binding, and signaling properties of CRF2(a) receptors endogenously expressed in human retinoblastoma Y79 cells: passage-dependent regulation of functional receptors

Eric Gutknecht, Richard L. Hauger, Ilse Van der Linden, Georges Vauquelin, Frank M. Dautzenberg

Journal:

Journal of Neurochemistry

Year:

2008

Language:

english

File:

PDF, 337 KB

english, 2008

18

Involvement of the AT1 receptor subtype in the effects of angiotensin IV and LVV-haemorphin 7 on hippocampal neurotransmitter levels and spatial working memory

Dimitri De Bundel, Heidi Demaegdt, Tony Lahoutte, Vicky Caveliers, Ken Kersemans, Ann-Gaelle Ceulemans, Georges Vauquelin, Ralph Clinckers, Patrick Vanderheyden, Yvette Michotte, Ilse Smolders

Journal:

Journal of Neurochemistry

Year:

2010

Language:

english

File:

PDF, 942 KB

english, 2010

19

Synergistic inhibition of the enzymatic activity of aminopeptidase N by divalent metal ion chelators

Patrick M.L. Vanderheyden, Heidi Demaegdt, Julie Swales, Pieter-Jan Lenaerts, Jean-Paul De Backer, Lotte K. Vogel, Georges Vauquelin

Journal:

Fundamental & Clinical Pharmacology

Year:

2006

Language:

english

File:

PDF, 564 KB

english, 2006

20

Unravelling the complex dissociation of [3H]-rimonabant from plated CB1 cannabinoid receptor-expressing cells

M. Wennerberg, A. Balendran, J.C. Clapham, Georges Vauquelin

Journal:

Fundamental & Clinical Pharmacology

Year:

2010

Language:

english

File:

PDF, 239 KB

english, 2010

21

Non-competitive interaction between raclopride and spiperone on human D2L-receptors in intact Chinese hamster ovary cells

Ann Packeu, Jean-Paul De Backer, Georges Vauquelin

Journal:

Fundamental & Clinical Pharmacology

Year:

2010

Language:

english

File:

PDF, 174 KB

english, 2010

22

Antagonist-D2S-dopamine receptors interactions in intact Chinese recombinant ovary cells

Ann Packeu, Tim Béghin, Jean-Paul De Backer, Georges Vauquelin

Journal:

Fundamental & Clinical Pharmacology

Year:

2010

Language:

english

File:

PDF, 250 KB

english, 2010

23

Binding properties of antagonists to Cannabinoid receptors in intact cells

Marie Wennerberg, Leifeng Cheng, Stephan Hjorth, John C. Clapham, Anudharan Balendran, Georges Vauquelin

Journal:

Fundamental & Clinical Pharmacology

Year:

2011

Language:

english

File:

PDF, 384 KB

english, 2011

24

Elusive equilibrium: the challenge of interpreting receptor pharmacology using calcium assays

Steven J Charlton, Georges Vauquelin

Journal:

British Journal of Pharmacology

Year:

2010

Language:

english

File:

PDF, 1.46 MB

english, 2010

25

Long-lasting target binding and rebinding as mechanisms to prolong in vivo drug action

Georges Vauquelin, Steven J Charlton

Journal:

British Journal of Pharmacology

Year:

2010

Language:

english

File:

PDF, 1.89 MB

english, 2010

26

Dopamine and Iron Induce Apoptosis in PC12 Cells

Carlos Velez-Pardo, Marlene Jimenez Del Rio, Hendrik Verschueren, Guy Ebinger, Georges Vauquelin

Journal:

Basic & Clinical Pharmacology & Toxicology

Year:

1997

Language:

english

File:

PDF, 1.19 MB

english, 1997

27

Identification of I1 and I2 Imidazoline Receptors in Striatum Membranes from Different Speciesa

GEORGES VAUQUELIN, JEAN-PAUL DE BACKER, PHILIPPE LADURE, ANJA FLAMEZ

Journal:

Annals of the New York Academy of Sciences

Year:

1999

File:

PDF, 808 KB

1999

28

Inhibition of Angiotensin II-Induced Inositol Phosphate Production by Triacid Nonpeptide Antagonists in CHO Cells Expressing Human AT1 Receptors

Patrick M. L. Vanderheyden, Ilse Verheijen, Frederik L. P. Fierens, Jean-Paul DeBacker, Georges Vauquelin

Journal:

Pharmaceutical Research

Year:

2000

Language:

english

File:

PDF, 174 KB

english, 2000

29

How can the differences among AT1-receptor antagonists Be explained?

Peter Morsing, Georges Vauquelin

Journal:

Cell Biochemistry and Biophysics

Year:

2001

Language:

english

File:

PDF, 149 KB

english, 2001

30

Amino Triazolo Diazepines (Ata) as Constrained Histidine Mimics

Buysse, Koen, Farard, Julien, Nikolaou, Alexandros, Vanderheyden, Patrick, Vauquelin, Georges, Sejer Pedersen, Daniel, Tourwé, Dirk, Ballet, Steven

Journal:

Organic Letters

Year:

2011

Language:

english

File:

PDF, 830 KB

english, 2011

31

Radioligand dissociation measurements: potential interference of rebinding and allosteric mechanisms and physiological relevance of the biological model systems

Vauquelin, Georges, Van Liefde, Isabelle

Journal:

Expert Opinion on Drug Discovery

Year:

2012

Language:

english

File:

PDF, 406 KB

english, 2012

32

Agonist-mediated conformational changes ofβ-adrenoceptors could occur independent of functional coupling to Ns

Yvonne Severne, Louis Kanarek, Georges Vauquelin

Journal:

Naunyn-Schmiedeberg's Archives of Pharmacology

Year:

1986

Language:

english

File:

PDF, 699 KB

english, 1986

33

Clozapine, atypical antipsychotics, and the benefits of fast-off D2dopamine receptor antagonism

Georges Vauquelin, Sophie Bostoen, Patrick Vanderheyden, Philip Seeman

Journal:

Naunyn-Schmiedeberg's Archives of Pharmacology

Year:

2012

Language:

english

File:

PDF, 981 KB

english, 2012

34

Serotonin binding proteins “SBP”: Target proteins and tool for in vitro neurotoxicity studies

Marlene Jimenez del Rio, Carlos Velez-Pardo, Guy Ebinger, Georges Vauquelin

Journal:

General Pharmacology: The Vascular System

Year:

1995

Language:

english

File:

PDF, 839 KB

english, 1995

35

Corrigendum

Hilde De Vos, Eva Czerwiec, Jean-Paul De Backer, Werner De Potter, Georges Vauquelin

Journal:

European Journal of Pharmacology: Molecular Pharmacology

Year:

1991

Language:

english

File:

PDF, 41 KB

english, 1991

36

Serotonin-binding proteins in the bovine cerebral cortex: interaction with serotonin and catecholamines

Marlene Jimenez Del Rio, Jef Pinxteren, Werner Do Potter, Guy Ebinger, Georges Vauquelin

Journal:

European Journal of Pharmacology: Molecular Pharmacology

Year:

1992

Language:

english

File:

PDF, 1.01 MB

english, 1992

37

Binding of serotonin and dopamine to ‘serotonin binding proteins’ in bovine frontal cortex: evidence for iron-induced oxidative mechanisms

Marlene Jimenez Del Rio, Carlos Velez Pardo, Jef Pinxteren, Werner De Potter, Guy Ebinger, Georges Vauquelin

Journal:

European Journal of Pharmacology: Molecular Pharmacology

Year:

1993

Language:

english

File:

PDF, 1.06 MB

english, 1993

38

Fe2+-mediated binding of serotonin and dopamine to skeletal muscle actin: resemblance to serotonin binding proteins

Carlos Velez Pardo, Marlen Jimenez del Rio, Jef Pinxteren, Werner De Potter, Guy Ebinger, Georges Vauquelin

Journal:

European Journal of Pharmacology: Molecular Pharmacology

Year:

1995

Language:

english

File:

PDF, 1.19 MB

english, 1995

39

Effect of saponin and filipin on antagonist binding to AT1 receptors in intact cells

Ilse Verheijen, Dieter Tourlousse, Patrick M.L Vanderheyden, Jean-Paul De Backer, Georges Vauquelin

Journal:

Biochemical Pharmacology

Year:

2004

Language:

english

File:

PDF, 196 KB

english, 2004

40

Synergistic modulation of cystinyl aminopeptidase by divalent cation chelators

Heidi Demaegdt, Hilde Laeremans, Jean-Paul De Backer, Sabrina Mosselmans, Minh Tam Le, Veerle Kersemans, Yvette Michotte, Georges Vauquelin, Patrick M.L Vanderheyden

Journal:

Biochemical Pharmacology

Year:

2004

Language:

english

File:

PDF, 189 KB

english, 2004

41

Endogenous cystinyl aminopeptidase in Chinese hamster ovary cells: characterization by [125I]Ang IV binding and catalytic activity

Heidi Demaegdt, Patrick Vanderheyden, Jean-Paul De Backer, Sabrina Mosselmans, Hilde Laeremans, Minh Tam Le, Veerle Kersemans, Yvette Michotte, Georges Vauquelin

Journal:

Biochemical Pharmacology

Year:

2004

Language:

english

File:

PDF, 184 KB

english, 2004

42

Cys2,7EtαCGRP is a potent agonist for CGRP1 receptors in SK-N-MC cells

Christina Nodin, Georges Vauquelin, Bengt von Mentzer

Journal:

Biochemical Pharmacology

Year:

2005

Language:

english

File:

PDF, 179 KB

english, 2005

43

Antagonist-radioligand binding to D2L-receptors in intact cells

Ann Packeu, Jean-Paul De Backer, Isabelle Van Liefde, Patrick M.L. Vanderheyden, Georges Vauquelin

Journal:

Biochemical Pharmacology

Year:

2008

Language:

english

File:

PDF, 377 KB

english, 2008

44

Involvement of insulin-regulated aminopeptidase and/or aminopeptidase N in the angiotensin IV-induced effect on dopamine release in the striatum of the rat

Bart Stragier, Heidi Demaegdt, Dimitri De Bundel, Ilse Smolders, Sophie Sarre, Georges Vauquelin, Guy Ebinger, Yvette Michotte, Patrick Vanderheyden

Journal:

Year:

2007

Language:

english

File:

PDF, 649 KB

english, 2007

45

KLHL12-mediated ubiquitination of the dopamine D4 receptor does not target the receptor for degradation

Pieter Rondou, Kamila Skieterska, Ann Packeu, Béatrice Lintermans, Peter Vanhoenacker, Georges Vauquelin, Guy Haegeman, Kathleen Van Craenenbroeck

Journal:

Cellular Signalling

Year:

2010

Language:

english

File:

PDF, 1012 KB

english, 2010

46

Ligand binding and functional properties of human angiotensin AT1 receptors in transiently and stably expressed CHO-K1 cells

Minh Tam Le, Jean-Paul De Backer, László Hunyady, Patrick M.L. Vanderheyden, Georges Vauquelin

Journal:

European Journal of Pharmacology

Year:

2005

Language:

english

File:

PDF, 467 KB

english, 2005

47

Angiotensin AT4 receptor ligand interaction with cystinyl aminopeptidase and aminopeptidase N: [125I]Angiotensin IV only binds to the cystinyl aminopeptidase apo-enzyme

Heidi Demaegdt, Pieter-Jan Lenaerts, Julie Swales, Jean-Paul De Backer, Hilde Laeremans, Minh Tam Le, Ken Kersemans, Lotte K. Vogel, Yvette Michotte, Patrick Vanderheyden, Georges Vauquelin

Journal:

European Journal of Pharmacology

Year:

2006

Language:

english

File:

PDF, 260 KB

english, 2006

48

Corticotropin-releasing factor receptors induce calcium mobilization through cross-talk with Gq-coupled receptors

Eric Gutknecht, Georges Vauquelin, Frank M. Dautzenberg

Journal:

European Journal of Pharmacology

Year:

2010

Language:

english

File:

PDF, 1.10 MB

english, 2010

49

Angiotensin II type 1 receptor antagonists: Why do some of them produce insurmountable inhibition?

Patrick M.L Vanderheyden, Frederik L.P Fierens, Georges Vauquelin

Journal:

Biochemical Pharmacology

Year:

2000

Language:

english

File:

PDF, 412 KB

english, 2000

50

A two-state receptor model for the interaction between angiotensin II type 1 receptors and non-peptide antagonists

Georges Vauquelin, Peter Morsing, Frederik L.P Fierens, Jean-Paul De Backer, Patrick M.L Vanderheyden

Journal:

Biochemical Pharmacology

Year:

2001

Language:

english

File:

PDF, 231 KB

english, 2001

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